Direct Asymmetric Reductive Amination for the Synthesis of (S)-Rivastigmine

Formal asymmetric biocatalytic reductive amination.

nano-rods zno as an efficient catalyst for the synthesis of chromene phosphonates, direct amidation and formylation of amines

چکیده ندارد.

Highly enantioselective hydrogen-transfer reductive amination: catalytic asymmetric synthesis of primary amines.

Optically active amines are attracting increasing interest in the food, agrochemical, and pharmaceutical industries as building blocks for novel compounds and as templates for asymmetric synthesis. One of the most common methods for preparing amines is the reductive amination of carbonyl compounds. We have successfully explored the rhodiumcatalyzed asymmetric reductive amination with hydrogen a...

Synthesis of chiral sultams via palladium-catalyzed intramolecular asymmetric reductive amination.

A novel palladium-catalyzed intramolecular reductive amination of ketones with weakly nucleophilic sulfonamides has been developed in the presence of a Brønsted acid, giving a wide range of chiral γ-, δ-, and ε-sultams in high yields and up to 99% of enantioselectivity.

Investigation of Reductive Amination in the Synthesis of T-0632

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